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Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50354485'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Inhibition human recombinant Abl using Abtide peptide substrate in presence of [gamma-32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Binding affinity to recombinant wild type human Abl using abitide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Binding affinity to human recombinant Abl by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed