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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase receptor UFO' and Ligand = 'BDBM50425829'
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataIC50:  3.99E+3nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused AXL (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human AXL by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed