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Found 9 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50378580'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-Urotensin-2 from human GPR14 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  5.01nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  0.832nMAssay Description:Agonist activity at urotensin-2 receptor in Sprague-Dawley rat aortic rings assessed as KCl-induced vasoconstrictionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed