Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a receptor' and Ligand = 'BDBM50052954'
TargetVasopressin V1a receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataIC50:  56nMAssay Description:Displacement of [3H]-AVP from AVP-V1a receptor binding site in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed