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Found 2 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor' and Ligand = 'BDBM50246609'
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246609((4R)-4-Ethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246609((4R)-4-Ethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-...)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed