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Found 2 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50329773'
TargetVesicular acetylcholine transporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50329773((-)-(2R,3R)-5-(2-fluoroethoxy)-3-(4-phenylpiperidi...)
Affinity DataKi:  19.6nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in rat PC12 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50329773((-)-(2R,3R)-5-(2-fluoroethoxy)-3-(4-phenylpiperidi...)
Affinity DataKi:  20nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed