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Found 2 Enz. Inhib. hit(s) with Target = 'Zinc metalloproteinase dpy-31' and Ligand = 'BDBM50063917'
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed