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Found 12 of ic50 for monomerid = 80396
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Dyrk1A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK4(Mus musculus)
University Of Kansas Specialized Chemistry Center

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  15nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK4 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Mus musculus)
University Of Kansas Specialized Chemistry Center

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  15nMAssay Description:Inhibition of mouse Clk4Checked by AuthorMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mouse Clk1Checked by AuthorMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mouse Clk1Checked by AuthorMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  20nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK1 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Mus musculus)
University Of Kansas Specialized Chemistry Center

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse recombinant GST-tagged CLK2 expressed in Escherichia coli DH5[alpha] using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH as substrate by l...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Mus musculus)
University Of Kansas Specialized Chemistry Center

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  200nMAssay Description:Inhibition of mouse Clk2Checked by AuthorMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  930nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA dC->dU-editing enzyme APOBEC-3A(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  2.69E+3nMT: 2°CAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA dC->dU-editing enzyme APOBEC-3G(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  2.89E+3nMT: 2°CAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDual specificity protein kinase CLK3(Mus musculus)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mouse Clk3Checked by AuthorMore data for this Ligand-Target Pair