Compile Data Set for Download or QSAR
maximum 50k data
Found 11 of ki for UniProtKB: P0AEK4
LigandPNGBDBM8726(5-chloro-2-(2,4-dichlorophenoxy)phenol | CHEMBL849...)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of wild type Escherichia coli FabI assessed as inhibition of bacterial growthMore data for this Ligand-Target Pair
LigandPNGBDBM36537(2-phenoxylphenol | PT51 | US10071965, Compound PT5...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of wild type Escherichia coli FabI assessed as inhibition of bacterial growthMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM36538(5-fluoro-2-phenoxylphenol | PT55 | US10071965, Com...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of wild type Escherichia coli FabI assessed as inhibition of bacterial growthMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM36539(5-chloro-2-phenoxylphenol | PT52 | US10071965, Com...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of wild type Escherichia coli FabI assessed as inhibition of bacterial growthMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM36542(5-methyl-2-phenoxylphenol | PT53 | US10071965, Com...)
Affinity DataKi:  7nMAssay Description:Inhibition of wild type Escherichia coli FabI assessed as inhibition of bacterial growthMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM190661(PT166)
Affinity DataKi:  7nMpH: 7.5Assay Description:Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 °C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...More data for this Ligand-Target Pair
LigandPNGBDBM231620(CG400549 | US10071965, Compound CG400549)
Affinity DataKi:  81.9nMpH: 7.5Assay Description:Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 °C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...More data for this Ligand-Target Pair
LigandPNGBDBM190652(LOX inhibitor, 13 | PT171)
Affinity DataKi:  95.7nMpH: 7.5Assay Description:Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 °C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM190654(PT173)
Affinity DataKi:  203nMpH: 7.5Assay Description:Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 °C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKi:  7.05E+3nMAssay Description:Inhibition of Escherichia coli MG1655 enoyl-ACP reductase overexpressed in Escherichia coli M15 assessed as oxidation of NADH to NAD+ after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of Escherichia coli MG1655 enoyl-ACP reductase overexpressed in Escherichia coli M15 assessed as oxidation of NADH to NAD+ after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed