Affinity DataIC50: 0.300nMAssay Description:In vivo binding affinity of the compound against dopamine (D1) receptor in rat caudate-putamen tissue using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.660nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]- #NAME? from binding Dopamine receptor D1 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.01nMAssay Description:Tested for its affinity towards Dopamine receptor D1 in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:In vivo binding affinity of the compound against dopamine (D1) receptor in rat caudate-putamen tissue using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Ability to inhibit binding of [3H]-SCH- 23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Ability to displace [3H]-SCH- 23390 (0.2 nM) from corpus striatum of rat Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]-SCH-23,390 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Compound was tested for binding affinity against dopamine Dopamine receptor D1 using 1 nM [3H]-SCH-23,390 as the radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2.15nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Ability to inhibit binding of [3H]-SCH- 23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Ability to inhibit binding of [3H]-SCH- 23390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Binding affinity towards dopamine receptor D1 by displacement of [3H]-SCH- radioligand in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Ability to displace [3H]-SCH- 23390 (0.2 nM) from corpus striatum of rat Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in Wistar rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Relative affinity for Dopamine receptor D1 in striatum using [3H]SCH-23390More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Displacement of [3H]-SCH- 23390 (0.3 nM) from dopamine receptor D1 in crude membrane fraction of rat brain corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Displacement of [3H]-SCH- 23390 (0.3 nM) from dopamine receptor D1 in crude membrane fraction of rat brain corpus striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Tested for its affinity towards Dopamine receptor D1 in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Binding affinity for dopamine receptor D1, activity is expressed as IC50 values.More data for this Ligand-Target Pair
Affinity DataIC50: 7.15nMAssay Description:Binding affinity against Dopamine receptor D1 by using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair