Compile Data Set for Download or QSAR
maximum 50k data
Found 26 of ic50 for UniProtKB: P67774
LigandPNGBDBM50110681(CHEMBL430266 | Calyculin-A)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135699((10S,13S,18S,19S,22R)-8-Isobutyl-18-((1E,3E)-(5S,6...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090505((1R,2S,6R,7S)-2,6-Dimethyl-4,10-dioxa-tricyclo[5.2...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at rat H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrsMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50556732(CHEMBL4750435)
Affinity DataIC50:  200nMAssay Description:Inhibition of PP2A alpha (unknown origin) pre-incubated for 20 mins followed by fluorescence substrate addition and measured after 120 mins by DiFMUP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50408821(CHEMBL5270968)
Affinity DataIC50:  400nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50135697(((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-methoxy-2,6...)
Affinity DataIC50:  500nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50453860(CHEMBL4210922)
Affinity DataIC50:  900nMAssay Description:Inhibition of recombinant human PP2A catalytic subunit L309 deletion mutant using DIFMUP as substrate pretreated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50135691((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135700((S)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135696((2R,5S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135687((R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135685((2S,5S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >3.90E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135683((2R,4R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135686((R)-2-((4E,6E)-(2S,3S)-3-Acetylamino-7-biphenyl-4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135689((2R,4R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135684((S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135688((R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135682((2S,4R)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135693((2R,4S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-m...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135690(CHEMBL98661 | [((4E,6E)-(2S,3S,8S,9S)-3-Acetylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135698((R)-2-((4E,6E)-(2S,3S)-3-Acetylamino-2,6-dimethyl-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135694((S)-1-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135692(CHEMBL100880 | N-[(2E,4E)-(1S,6S,7S)-7-Methoxy-4,6...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50135695((R)-2-[(4E,6E)-(2S,3S)-3-Acetylamino-7-(2-benzyl-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed