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Found 3 of ec50 for UniProtKB: P33766
TargetfMet-Leu-Phe receptor(Mus musculus)TBA
LigandPNGBDBM50559829(CHEMBL4784510)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at mouse FPR1 expressed in CHO-A12 cells assessed as cAMP level incubated for 1.5 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetfMet-Leu-Phe receptor(Mus musculus)TBA
LigandPNGBDBM50186957(1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse FPR1 expressed in CHO-A12 cells assessed as cAMP level incubated for 1.5 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetfMet-Leu-Phe receptor(Mus musculus)TBA
LigandPNGBDBM50559829(CHEMBL4784510)
Affinity DataEC50:  500nMAssay Description:Agonist activity at mouse FPR1 expressed in CHO cells assessed as reduction cAMP accumulation incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed