Compile Data Set for Download or QSAR
maximum 50k data
Found 26 of ic50 for UniProtKB: P30897
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212643(CHEMBL308516)
Affinity DataIC50:  2.25nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  2.33nMAssay Description:Tested for the inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  3.57nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212634(CHEMBL309009)
Affinity DataIC50:  5.23nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212636(CHEMBL310221)
Affinity DataIC50:  7.55nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212635(CHEMBL415266)
Affinity DataIC50:  7.61nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212645(CHEMBL305908)
Affinity DataIC50:  7.91nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212646(CHEMBL72972)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212638(CHEMBL302512)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212644(CHEMBL73450)
Affinity DataIC50:  25.5nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212637(CHEMBL72046)
Affinity DataIC50:  37.1nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  37.5nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  65.3nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212639(CHEMBL302241)
Affinity DataIC50:  72.4nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  95.4nMAssay Description:Inhibition of Proteus mirabilis C889 beta-lactamase assessed as inhibition of nitrocefin hydrolysis preincubated for 5 mins by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  342nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50021959(CHEMBL777 | MM 14151 | US9120808, Clavulanic acid ...)
Affinity DataIC50:  9.54E+4nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469657(CHEMBL33995 | SB-202742)
Affinity DataIC50:  2.99E+5nMAssay Description:Inhibition of Proteus mirabilis C889 beta-lactamase assessed as inhibition of nitrocefin hydrolysis preincubated for 5 mins by microtiter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469666(6-Octylsalicylic Acid | CHEMBL33379)
Affinity DataIC50:  1.55E+7nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469665(CHEMBL30914)
Affinity DataIC50:  2.20E+7nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469660(CHEMBL30915)
Affinity DataIC50:  6.06E+7nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50:  9.05E+7nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469657(CHEMBL33995 | SB-202742)
Affinity DataIC50:  2.96E+8nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469661(CHEMBL30870)
Affinity DataIC50:  6.15E+8nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50469667(6-Decylsalicylic Acid | CHEMBL416038)
Affinity DataIC50:  6.46E+8nMAssay Description:Concentration required for its inhibitory activity against Proteus mirabilis C889 class A beta-lactamaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article