Affinity DataKi: 0.600nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro inhibition constant for Aurora-CMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:In vitro inhibition constant for Aurora-BMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro inhibition constant for FLT-3More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: <1nMAssay Description:Inhibition of Aurora A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of in vitro Aurora-B kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of in vitro Aurora-A kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of Aurora-B immunoprecipitated from mitotic cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 452nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 472nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 483nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 578nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against EGFRMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition constant for Aurora-AMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against SRCMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against FGFRMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against human hERG receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of in vitro Plk1 kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of in vitro CDK1 kinase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against IGFRMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against CSKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against JAK3More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibitory activity against CDK2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against p38-alpha MAPKMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against JNK1alphaMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit alpha/beta/gamma(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PKAMore data for this Ligand-Target Pair