Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with all data for assayid = 5 entry = 50035536
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027041(2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...)
Affinity DataKi:  120nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  1.24E+3nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50046325((S)-2-((2S,3S)-3-Amino-2-hydroxy-4-phenyl-butyryla...)
Affinity DataKi:  1.70E+4nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataKi:  2.00E+4nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027049(2-(3-Amino-2-methyl-4-phenyl-butyrylamino)-4-methy...)
Affinity DataKi:  3.78E+6nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed