Compile Data Set for Download or QSAR
maximum 50k data
Found 134 Enz. Inhib. hit(s) with all data for entry = 50018615
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197470((1S,2S,3S,7R)-methyl 3-(3,4-dichlorophenyl)-7-hydr...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197437((1R,2S,3R)-methyl 3-(3,4-dichlorophenyl)-8-methyl-...)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197441((1S,2S,3R,7R)-methyl 3-(3,4-dichlorophenyl)-7-hydr...)
Affinity DataIC50:  0.760nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197469((1R,2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197452((1R)-methyl 3-(3,4-dichlorophenyl)-8-methyl-8-aza-...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197477((1R)-2-beta-carbomethoxy-3-beta-(3,4-dichloropheny...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197456((1R,2S,3R)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bic...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197453((1R)-2-carbomethoxy-3-(3,4-dichlorophenyl)-8-thiab...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197469((1R,2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-methyl-...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197477((1R)-2-beta-carbomethoxy-3-beta-(3,4-dichloropheny...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197457((2S,3R)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197486((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197443((1R,2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bic...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50156398(2-carbomethoxy-3-(3,4-dichlorophenyl)-8-thiabicycl...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197458((1R)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicyclo[3...)
Affinity DataIC50:  4.60nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197443((1R,2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bic...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197460((1R)-2-beta-carbomethoxy-3-alpha-(3,4-dichlorophen...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197448((1S)-2-carbomethoxy-3-(3,4-dichlorophenyl)-8-thiab...)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197438(2-beta-carbomethoxy-3-beta-(3,4-dichlorophenyl)-8-...)
Affinity DataIC50:  5.30nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197471((2R,3S)-methyl 3-(3,4-dichlorophenyl)-8-thia-bicyc...)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197462(2-beta-carbomethoxy-3-beta-(4-bromophenyl)-8-thiab...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197491(2-beta-carbomethoxy-3-beta-(4-chloro-3-fluoropheny...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197474(2-beta-carbomethoxy-3-alpha-(4-bromophenyl)-8-thia...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197486((2S,3S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  6.5nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197449(2-beta-carbomethoxy-3-beta-(3-chloro-4-fluoropheny...)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50156395(2-carbomethoxy-3-(4-iodophenyl)-8-thiabicyclo-[3.2...)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197440(2-beta-carbomethoxy-3-alpha-(3,4-dichlorophenyl)-8...)
Affinity DataIC50:  6.90nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197447(2-beta-carbomethoxy-3-alpha-(4-chloro-3-fluorophen...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197450(2-beta-carbomethoxy-3-alpha-(3-chloro-4-fluorophen...)
Affinity DataIC50:  7.10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50076048((1R/1S)-methyl 3-(3,4-dichlorophenyl)bicyclo[3.2.1...)
Affinity DataIC50:  7.10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197476((1S,7R)-methyl 3-(3,4-dichlorophenyl)-7-hydroxy-8-...)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197490(2-carbomethoxy-3-(3-chloro-4-fluorophenyl)-8-thiab...)
Affinity DataIC50:  7.60nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197446(2-beta-carbomethoxy-3-alpha-(3,4-dichlorophenyl)-8...)
Affinity DataIC50:  7.80nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50156401(2-carbomethoxy-3-(2-naphthyl)-8-thiabicyclo-[3.2.1...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197471((2R,3S)-methyl 3-(3,4-dichlorophenyl)-8-thia-bicyc...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197492(2-beta-carbomethoxy-3-alpha-(2-naphthyl)-8-thiabic...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197451(2-beta-carbomethoxy-3-alpha-(4-iodophenyl)-8-thiab...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50156391(2-carbomethoxy-3-(4-bromophenyl)-8-thiabicyclo-[3....)
Affinity DataIC50:  9.10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197436((2R,3S)-methyl 3-(3,4-dichlorophenyl)bicyclo[3.2.1...)
Affinity DataIC50:  9.60nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197445(2-beta-carbomethoxy-3-beta-(4-chlorophenyl)-8-thia...)
Affinity DataIC50:  9.60nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197466(2-carbomethoxy-3-(4-chloro-3-fluorophenyl)-8-thiab...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197481(2-beta-carbomethoxy-3-beta-(4-iodophenyl)-8-thiabi...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197444((1S)-2-beta-carbomethoxy-3-alpha-(3,4-dichlorophen...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50076047((1R/1S)-methyl 3-(3,4-dichlorophenyl)-8-oxa-bicycl...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197465(2-beta-carbomethoxy-3alpha-(4-chlorophenyl)-8-thia...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197488(2-beta-carbomethoxy-3-alpha-(3,4-difluorophenyl)-8...)
Affinity DataIC50:  11.3nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197472((2R,3R)-methyl 3-(3,4-dichlorophenyl)bicyclo[3.2.1...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50156390(2-carbomethoxy-3-(4-chlorophenyl)-8-thiabicyclo-[3...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Macaca mulatta)
Organix

Curated by ChEMBL
LigandPNGBDBM50197439(2-beta-carbomethoxy-3-beta-(2-naphthyl)-8-thiabicy...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]citalopram from SERT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50197481(2-beta-carbomethoxy-3-beta-(4-iodophenyl)-8-thiabi...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]WIN 35428 from DAT in rhesus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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