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Found 78 Enz. Inhib. hit(s) with all data for entry = 50033177
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340942(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(n...)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  40nMAssay Description:Inhibition of VEGFR-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340939(CHEMBL1761939 | N-(3-chloro-4-fluorophenyl)-N'-{4-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340937(1-(4-bromophenyl)-3-(4-(6,7-dimethoxyquinazolin-4-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340941(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-pa...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340940(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(4...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340929(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-ph...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM3032(CHEMBL1204168 | CHEMBL29197 | N-(3-bromophenyl)-6,...)
Affinity DataIC50:  63nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50162157(1-[4-(6,7-Dimethoxy-quinazolin-4-yloxy)-phenyl]-3-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50162157(1-[4-(6,7-Dimethoxy-quinazolin-4-yloxy)-phenyl]-3-...)
Affinity DataIC50:  70nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340938(1-(2,4-difluorophenyl)-3-(4-(6,7-dimethoxyquinazol...)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340936(1-butyl-3-(4-(6,7-dimethoxyquinazolin-4-yloxy)phen...)
Affinity DataIC50:  400nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  500nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340933(1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-ph...)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340926(CHEMBL1761932 | ethyl 4-(6,7-dimethoxyquinazolin-4...)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340920(4-(4-bromo-2-fluorophenoxy)-6,7-dimethoxyquinazoli...)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340935(1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(4...)
Affinity DataIC50:  600nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340924(CHEMBL1761930 | methyl 4-(6,7-dimethoxyquinazolin-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50184861(CHEMBL205089 | N-Cyclohexyl-N'-{4-[6,7-dimethoxy-4...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340918(4-(4-Bromo-2-fluoroanilino)-6,7-dimethoxyquinazoli...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340944(1-(3-chloro-4-fluorophenyl)-3-(4-(6,7-dimethoxyqui...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340927(1-(4-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-3-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340943(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(n...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340925(CHEMBL1761931 | Ethyl {4-[6,7-dimethoxy-quinazolin...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340918(4-(4-Bromo-2-fluoroanilino)-6,7-dimethoxyquinazoli...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340923(CHEMBL1761929 | Methyl {4-[6,7-dimethoxy-quinazoli...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340920(4-(4-bromo-2-fluorophenoxy)-6,7-dimethoxyquinazoli...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340930(1-(4-(6,7-dimethoxyquinazolin-4-ylamino)phenyl)-3-...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340923(CHEMBL1761929 | Methyl {4-[6,7-dimethoxy-quinazoli...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50290838(4-(3-Bromo-phenoxy)-6,7-dimethoxy-quinazoline | CH...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340917(4-(3-chloro-4-fluorophenoxy)-6,7-dimethoxyquinazol...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50290838(4-(3-Bromo-phenoxy)-6,7-dimethoxy-quinazoline | CH...)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of recombinant human VEGFR-2-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340932(1-(3-((6,7-dimethoxyquinazolin-4-yl)(methyl)amino)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340933(1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340934(1-(3-((6,7-dimethoxyquinazolin-4-yl)(methyl)amino)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340935(1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340936(1-butyl-3-(4-(6,7-dimethoxyquinazolin-4-yloxy)phen...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340937(1-(4-bromophenyl)-3-(4-(6,7-dimethoxyquinazolin-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340938(1-(2,4-difluorophenyl)-3-(4-(6,7-dimethoxyquinazol...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340939(CHEMBL1761939 | N-(3-chloro-4-fluorophenyl)-N'-{4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340941(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-pa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340942(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(n...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340943(1-(4-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(n...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50184861(CHEMBL205089 | N-Cyclohexyl-N'-{4-[6,7-dimethoxy-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50340944(1-(3-chloro-4-fluorophenyl)-3-(4-(6,7-dimethoxyqui...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human EGFR-mediated poly(Glu4Tyr) phosphorylation after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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