Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+4nMAssay Description:Inhibition of APN in human HL60 cells assessed as hydrolysis of L-Leu-p-nitroanilide by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of APN in human HL60 cells assessed as hydrolysis of L-Leu-p-nitroanilide by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.04E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.22E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.22E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4.41E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 5.27E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.13E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.32E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.63E+4nMAssay Description:Inhibition of APN in human HL60 cells assessed as hydrolysis of L-Leu-p-nitroanilide by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.74E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7.47E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.06E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.39E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.43E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.66E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+5nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair