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Found 46 Enz. Inhib. hit(s) with all data for entry = 50029714
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50071960(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  8nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287178(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  24nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  24nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287176(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  39nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287175(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  40nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287163(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  50nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287173(4-Chloro-1-methoxy-naphthalene-2-carboxylic acid [...)
Affinity DataKi:  55nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287165(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  66nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287179(4-Cyano-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  71nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287168(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  76nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287179(4-Cyano-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  131nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287180(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  132nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287178(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  151nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287169(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  260nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287164(4-Bromo-1-ethoxy-naphthalene-2-carboxylic acid [2-...)
Affinity DataKi:  267nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287170(1-Methoxy-naphthalene-2-carboxylic acid [2-(4-phen...)
Affinity DataKi:  270nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287168(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  303nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287167(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  339nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287165(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  484nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287176(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  517nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287166(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  652nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287162(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  652nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287175(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  703nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287177(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  731nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287174(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  731nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287169(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  996nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287163(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287167(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  1.21E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287166(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  1.29E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287162(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  1.29E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  1.89E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287173(4-Chloro-1-methoxy-naphthalene-2-carboxylic acid [...)
Affinity DataKi:  2.53E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287177(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  5.69E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287174(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataKi:  5.69E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287170(1-Methoxy-naphthalene-2-carboxylic acid [2-(4-phen...)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287164(4-Bromo-1-ethoxy-naphthalene-2-carboxylic acid [2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287171(4-Bromo-naphthalene-2-carboxylic acid [2-(4-phenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287171(4-Bromo-naphthalene-2-carboxylic acid [2-(4-phenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287172(4-Bromo-1-hydroxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287172(4-Bromo-1-hydroxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287176(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataEC50:  83nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287163(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataEC50:  68nMAssay Description:Compound was evaluated for effective concentration required for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50071960(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataEC50:  13nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataEC50:  68nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287175(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2...)
Affinity DataEC50:  28nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287165(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataEC50: >1.00E+3nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article