Affinity DataKi: 44nMAssay Description:Compound was evaluated for inhibitory activity against [3H]-BK in membrane preparations from a stable cell line that expresses the human B2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Compound was evaluated for inhibitory activity against [3H]-BK in the classical guinea pig ileum B2 binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 980nMAssay Description:Compound was evaluated for agonist activity against B1 receptor in rat ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 85nMAssay Description:Functional antagonism against BK-induced contractions in the classical guinea pig ileum B2 binding assayMore data for this Ligand-Target Pair