Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50030043
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214791(CHEMBL3142597)
Affinity DataKi:  44nMAssay Description:Compound was evaluated for inhibitory activity against [3H]-BK in membrane preparations from a stable cell line that expresses the human B2 receptorMore data for this Ligand-Target Pair
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TargetB2 bradykinin receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50214793(CHEMBL3142595)
Affinity DataKi:  360nMAssay Description:Compound was evaluated for inhibitory activity against [3H]-BK in the classical guinea pig ileum B2 binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetB1 bradykinin receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50290545((S)-2-{[(S)-1-((S)-2-{13-[(S)-2-((S)-2,6-Diamino-h...)
Affinity DataEC50:  980nMAssay Description:Compound was evaluated for agonist activity against B1 receptor in rat ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails Article
TargetB1 bradykinin receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50214792(CHEMBL264100 | des-Arg10-Kallidin)
Affinity DataEC50:  85nMAssay Description:Functional antagonism against BK-induced contractions in the classical guinea pig ileum B2 binding assayMore data for this Ligand-Target Pair
In DepthDetails Article