Reaction Details Report a problem with these data
Target
Serine/threonine-protein kinase 17B
Ligand
BDBM50509370
Substrate
n/a
Meas. Tech.
ChEMBL_1838143 (CHEMBL4338276)
IC50
8300±n/a nM
Citation
Hansen, KØ; Andersen, JH; Bayer, A; Pandey, SK; Lorentzen, M; Jørgensen, KB; Sydnes, MO; Guttormsen, Y; Baumann, M; Koch, U; Klebl, B; Eickhoff, J; Haug, BE; Isaksson, J; Hansen, EH Kinase Chemodiversity from the Arctic: The Breitfussins. J Med Chem 62:10167-10181 (2019) [PubMed] Article
More Info.:
Target
Name:
Serine/threonine-protein kinase 17B
Synonyms:
DRAK2 | ST17B_HUMAN | STK17B | Serine/threonine-protein kinase 17B | Serine/threonine-protein kinase 17B (STK17B)
Type:
Enzyme
Mol. Mass.:
42332.49
Organism:
Homo sapiens (Human)
Description:
O94768
Residue:
372
Sequence:
MSRRRFDCRSISGLLTTTPQIPIKMENFNNFYILTSKELGRGKFAVVRQCISKSTGQEYAAKFLKKRRRGQDCRAEILHEIAVLELAKSCPRVINLHEVYENTSEIILILEYAAGGEIFSLCLPELAEMVSENDVIRLIKQILEGVYYLHQNNIVHLDLKPQNILLSSIYPLGDIKIVDFGMSRKIGHACELREIMGTPEYLAPEILNYDPITTATDMWNIGIIAYMLLTHTSPFVGEDNQETYLNISQVNVDYSEETFSSVSQLATDFIQSLLVKNPEKRPTAEICLSHSWLQQWDFENLFHPEETSSSSQTQDHSVRSSEDKTSKSSCNGTCGDREDKENIPEDSSMVSKRFRFDDSLPNPHELVSDLLC