Reaction Details Report a problem with these data
Target
Gelatinase
Ligand
BDBM634009
Substrate
n/a
Meas. Tech.
Inhibition of Collagenase H Assay
IC50
1690±n/a nM
Citation
HOEKSTRA, W; RYU, H; CHINTHA, P SMALL MOLECULE INHIBITORS OF BACTERIAL TOXINS US Patent US20230357139 Publication Date 11/9/2023
More Info.:
Target
Name:
Gelatinase
Synonyms:
Coccolysin
Type:
Protein
Mol. Mass.:
55485.95
Organism:
n/a
Description:
Q833V7
Residue:
510
Sequence:
MMKGNKILYILGTGIFVGSSCLFSSLFVAAEEQVYSESEVSTVLSKLEKEAISEAAAEQYTVVDRKEDAWGMKHLKLEKQTEGVTVDSDNVIIHLDRNGAVTSVTGNPVDQVVKIQSVDAIGEEGVKKIIASDNPETKDLVFLAIDKRVNNEGQLFYKVRVTSSPTGDPVSLVYKVNATDGTIMEKQDLTEHVGSEVTLKNSFQVAFNVPVEKSNTGIALHGTDNTGVYHAVVDGKNNYSIIQAPSLVALNQNAVDAYTHGKFVKTYYEDHFQRHSIDDRGMPILSVVDEQHPDAYDNAFWDGKAMRYGETSTPTGKTYASSLDVVGHEMTHGVTEHTAGLEYLGQSGALNESYSDLMGYIISGASNPEIGADTQSVDRKTGIRNLQTPSKHGQPETMAQYDDRARYKGTPYYDQGGVHYNSGIINRIGYTIIQNLGIEKAQTIFYSSLVNYLTPKAQFSDARDAMLAAAKVQYGDEAASVVSAAFNSAGIGAKEDIQVNQPSESVLVNE