Compile Data Set for Download or QSAR
Report error Found 34 of affinity data for UniProtKB/TrEMBL: O54814
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163636BDBM50163636(1-((1R,2S)-2-(((S)-3-(4-fluorobenzyl)piperidin-1-y...)
Affinity DataIC50: 0.00700nMAssay Description:Inhibition of eotaxin-induced chemotaxis of rat eosinophilsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50163634BDBM50163634(1-{(1R,2S)-2-[(S)-3-(4-Fluoro-benzyl)-piperidin-1-...)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of eotaxin-induced chemotaxis of rat eosinophilsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041183BDBM50041183(CHEMBL3355941)
Affinity DataKi:  100nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041174BDBM50041174(CHEMBL3355938)
Affinity DataKi:  260nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041190BDBM50041190(CHEMBL3355951)
Affinity DataKi:  260nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041150BDBM50041150(CHEMBL3355932)
Affinity DataKi:  260nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041090BDBM50041090(CHEMBL3355964)
Affinity DataKi:  320nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041088BDBM50041088(CHEMBL3355962)
Affinity DataKi:  390nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041186BDBM50041186(CHEMBL3355945)
Affinity DataKi:  420nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041187BDBM50041187(CHEMBL3355946)
Affinity DataKi:  560nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041191BDBM50041191(CHEMBL3355952)
Affinity DataKi:  560nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041158BDBM50041158(CHEMBL3355934)
Affinity DataKi:  630nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041181BDBM50041181(CHEMBL3355939)
Affinity DataKi:  730nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041157BDBM50041157(CHEMBL3355933)
Affinity DataKi:  880nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041166BDBM50041166(CHEMBL3355936)
Affinity DataKi:  950nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041089BDBM50041089(CHEMBL3355963)
Affinity DataKi:  990nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041185BDBM50041185(CHEMBL3355944)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041195BDBM50041195(CHEMBL3355956)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041193BDBM50041193(CHEMBL3355954)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041182BDBM50041182(CHEMBL3355940)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041198BDBM50041198(CHEMBL3355960)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041189BDBM50041189(CHEMBL3355949)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041163BDBM50041163(CHEMBL3355935)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041194BDBM50041194(CHEMBL3355955)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50161407BDBM50161407([(3S,4S)-4-(3,4-Dichloro-benzyl)-3-hydroxymethyl-[...)
Affinity DataKi:  2.98E+3nMAssay Description:In vitro binding affinity against rat CC chemokine receptor 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041092BDBM50041092(CHEMBL3355966)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041091BDBM50041091(CHEMBL3355965)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041188BDBM50041188(CHEMBL3355947)
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041167BDBM50041167(CHEMBL3355937)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041184BDBM50041184(CHEMBL3355943)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041196BDBM50041196(CHEMBL3355958)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041197BDBM50041197(CHEMBL3355959)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041192BDBM50041192(CHEMBL3355953)
Affinity DataKi:  5.50E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetC-C chemokine receptor type 3(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041199BDBM50041199(CHEMBL3355961)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [125J]-eotaxin-1 from rat CCR3 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed