Affinity DataIC50: 0.200nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:In vitro binding affinity of the compound towards rat glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Compound was evaluated in vitro for its inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Compound was tested for its ability to displace [I-125]-glucagon from the glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagon (inactive up to 100 microM)More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 21.2nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity of the compound towards rat Glucagon ReceptorMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
Affinity DataIC50: 34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:pA2 value towards glucagon receptor relative to glucagon was calculatedMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 85nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 101nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 113nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair