Compile Data Set for Download or QSAR
maximum 50k data
Found 117 of affinity data for UniProtKB/TrEMBL: P30082
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104037(CHEMBL428460 | His-Ser-Gln-Gly-Lys-Phe-Thr-Ser-Glu...)
Affinity DataIC50:  0.200nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104040(CHEMBL412488 | His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp...)
Affinity DataIC50:  0.240nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataIC50:  0.430nMAssay Description:In vitro binding affinity of the compound towards rat glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50:  1nMAssay Description:Compound was evaluated in vitro for its inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(CHEMBL429362 | His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:Compound was tested for its ability to displace [I-125]-glucagon from the glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104030(CHEMBL439885 | His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp...)
Affinity DataIC50:  1.70nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051586(CHEMBL413666 | [des-His1,Tyr5,Glu9,D-Tyr10]glucago...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104039(CHEMBL267189 | His-Ser-Gln-Cys-Thr-Phe-Thr-Ser-Cys...)
Affinity DataIC50:  3.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098563(CHEMBL413890 | Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr...)
Affinity DataIC50:  3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407844(CHEMBL2115191)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104031(CHEMBL263603 | His-Cys-Gln-Gly-Thr-Phe-Cys-Ser-Asp...)
Affinity DataIC50:  5.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104043(CHEMBL437648 | His-Ser-Lys-Gly-Thr-Phe-Glu-Ser-Asp...)
Affinity DataIC50:  6nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104041(CHEMBL414077 | His-Ser-Gln-Gly-Thr-Phe-Cys-Ser-Asp...)
Affinity DataIC50:  6.40nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50454201(CHEMBL3037804)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104033(CHEMBL442135 | His-Ser-Gln-Gly-Thr-Phe-Lys-Ser-Asp...)
Affinity DataIC50:  14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104044(CHEMBL409654 | His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp...)
Affinity DataIC50:  14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098573(CHEMBL267876 | N-trinitrophenyl-His-Ser-Gln-Gly-Th...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagon (inactive up to 100 microM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352(CHEMBL442499 | [des-His1, Trp6, Glu9] glucagon-NH2)
Affinity DataIC50:  19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098566(CHEMBL413208 | phenylbutyryl-Tyr-Ser-Lys-Tyr-Leu-A...)
Affinity DataIC50:  21.2nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50:  23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50:  27nMAssay Description:Binding affinity of the compound towards rat Glucagon ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098572(Ac-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg...)
Affinity DataIC50:  31nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50407842(CHEMBL2114176)
Affinity DataIC50:  34.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  36nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358(CHEMBL267885 | [des-His1, Tyr6,Glu9] glucagon-NH2)
Affinity DataIC50:  40nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50244455((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...)
Affinity DataIC50:  43nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356(CHEMBL2369990 | [des-His1, Nle6, Glu9] glucagon-NH...)
Affinity DataIC50:  48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098570(CHEMBL438045 | Ser-Gln-Gly-Thr-Thr-Ser-Glu-Tyr-Ser...)
Affinity DataIC50:  48nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362(CHEMBL268636 | [des-His1, des-Phe6, Glu9] glucagon...)
Affinity DataIC50:  48nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50284992(CHEMBL441209 | H-Ser-Gln-GlyThr-Thr-Ser-Glu-Tyr-Se...)
Affinity DataIC50:  48nMAssay Description:pA2 value towards glucagon receptor relative to glucagon was calculatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359(CHEMBL411289 | [des-His1, des-Gly4, Glu9] glucagon...)
Affinity DataIC50:  52nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50087848(CHEMBL427644 | c[Asp15, Lys18,] glucagon-NH2)
Affinity DataIC50:  54nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50144009(3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluorome...)
Affinity DataIC50:  56nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098565(Ac-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50:  60nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50051585(CHEMBL2369127 | [des-His1,Tyr5,Glu9,(2S,3R)-beta-M...)
Affinity DataIC50:  74nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104036(CHEMBL414490 | His-Ser-Gln-Cys-Thr-Phe-Thr-Ser-Cys...)
Affinity DataIC50:  85nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50057824(CHEMBL3326175)
Affinity DataIC50:  87nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059364(CHEMBL2369985 | [des-His1, D-Phe6, Glu9] glucagon-...)
Affinity DataIC50:  100nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50104032(CHEMBL441011 | His-Cys-Gln-Gly-Thr-Phe-Cys-Ser-Asp...)
Affinity DataIC50:  101nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059365(CHEMBL412352 | [des-Phe6, Glu9] glucagon-NH2)
Affinity DataIC50:  113nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50:  122nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059363(CHEMBL437095 | [des-His1,Ala6, Glu9] glucagon-NH2)
Affinity DataIC50:  126nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50059360(CHEMBL429198 | [des-His1, des-Phe6] glucagon-NH2)
Affinity DataIC50:  128nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50087843(CHEMBL429724 | c[Asp9, Lys12,] glucagon-NH2)
Affinity DataIC50:  130nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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