TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.60E+5nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.70E+5nMAssay Description:Compound was tested for the binding affinity towards muscarinic receptor in mouse brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Compound was tested for the competitive inhibition of phosphonylation of Eel acetylcholinesterase (AChE)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKd: 9.10E+3nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 9.90E+3nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKd: 1.50E+4nMAssay Description:In vitro inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKd: 2.50E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKd: 1.40E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Mus musculus)
Sri International
Curated by ChEMBL
Sri International
Curated by ChEMBL
Affinity DataKd: 7.00E+4nMAssay Description:Displacement of [3H]5-HT binding to serotonin receptor of rat fundus membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80E+3nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Tested against Muscarinic acetylcholine receptor M3 expressed in A9 L cell lineMore data for this Ligand-Target Pair