Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 12810
TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730174(US12264155, Compound 61)
Affinity DataIC50: 2nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730186(US12264155, Compound 73)
Affinity DataIC50: 3nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730119(US12264155, Compound 5)
Affinity DataIC50: 3nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730142(US12264155, Compound 28)
Affinity DataIC50: 4nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730203(US12264155, Compound 91)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730184(US12264155, Compound 71)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730169(US12264155, Compound 56)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730198(US12264155, Compound 86)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730183(US12264155, Compound 70)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730161(US12264155, Compound 48)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730190(US12264155, Compound 77)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730159(US12264155, Compound 45)
Affinity DataIC50: 5nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730138(US12264155, Compound 24)
Affinity DataIC50: 6nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730171(US12264155, Compound 58)
Affinity DataIC50: 6nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730193(US12264155, Compound 80)
Affinity DataIC50: 6nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730204(US12264155, Compound 92)
Affinity DataIC50: 8nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730187(US12264155, Compound 74)
Affinity DataIC50: 8nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730165(US12264155, Compound 52)
Affinity DataIC50: 8nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730194(US12264155, Compound 81)
Affinity DataIC50: 8nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730166(US12264155, Compound 53)
Affinity DataIC50: 9nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730197(US12264155, Compound 84)
Affinity DataIC50: 9nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730117(US12264155, Compound 3)
Affinity DataIC50: 9nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730172(US12264155, Compound 59)
Affinity DataIC50: 10nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730157(US12264155, Compound 43)
Affinity DataIC50: 10nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730199(US12264155, Compound 87)
Affinity DataIC50: 10nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730170(US12264155, Compound 57)
Affinity DataIC50: 11nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730162(US12264155, Compound 49)
Affinity DataIC50: 11nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730176(US12264155, Compound 63)
Affinity DataIC50: 11nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730160(US12264155, Compound 47)
Affinity DataIC50: 12nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730168(US12264155, Compound 55)
Affinity DataIC50: 13nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730195(US12264155, Compound 82)
Affinity DataIC50: 17nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730175(US12264155, Compound 62)
Affinity DataIC50: 19nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730196(US12264155, Compound 83)
Affinity DataIC50: 22nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730167(US12264155, Compound 54)
Affinity DataIC50: 23nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730191(US12264155, Compound 78)
Affinity DataIC50: 24nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730158(US12264155, Compound 44)
Affinity DataIC50: 27nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730188(US12264155, Compound 75)
Affinity DataIC50: 29nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730200(US12264155, Compound 88)
Affinity DataIC50: 30nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730192(US12264155, Compound 79)
Affinity DataIC50: 30nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730201(US12264155, Compound 89)
Affinity DataIC50: 31nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730156(US12264155, Compound 42)
Affinity DataIC50: 32nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730189(US12264155, Compound 76)
Affinity DataIC50: 36nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730173(US12264155, Compound 60)
Affinity DataIC50: 37nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730123(US12264155, Compound 9)
Affinity DataIC50: 37nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730116(US12264155, Compound 2)
Affinity DataIC50: 40nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730146(US12264155, Compound 32)
Affinity DataIC50: 54nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730118(US12264155, Compound 4)
Affinity DataIC50: 56nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM729984(US12264155, Compound 1)
Affinity DataIC50: 57nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730177(US12264155, Compound 64)
Affinity DataIC50: 92nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetSerine/threonine-protein kinase ATR(Human)
Repare Therapeutics

US Patent
LigandPNGBDBM730185(US12264155, Compound 72)
Affinity DataIC50: 94nMAssay Description:Detection of ATR kinase activity utilized the AlphaScreen system to measure the phosphorylation of the substrate protein p53. Recombinant purified AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

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