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Found 347 with Last Name = 'avery' and Initial = 'ma'
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303975(3'-(4-(2-(1H-Tetrazol-5-yl)ethyl)benzyl)-1,7'-dime...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi:  390nMAssay Description:Binding affinity to 5HT2B receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi:  560nMAssay Description:Binding affinity to sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303976(3'-(2-(4-(2-(1H-Tetrazol-5-yl)ethyl)phenoxy)ethyl)...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303977(3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'-biben...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303979(CHEMBL571763 | Ethyl 3-(4-(2-(1,7'-Dimethyl-2'-pro...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303978(1-(4-(2-(1H-tetrazol-5-yl)ethyl)benzyl)-4-methyl-2...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303980(1-(4-((1H-Tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataKi:  5.06E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303986(CHEMBL584704 | Ethyl 2-Methyl-3-(4-(2-(4-methyl-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adrenoceptor alpha 2B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens)
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adrenoceptor alpha 2A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adrenoceptor alpha 1B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adrenoceptor alpha 1A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to beta1 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adrenoceptor alpha 2C (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to dopamine D5 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to histamine H3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to histamine H4 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to muscarinic acetylcholine receptor M2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to muscarinic acetylcholine receptor M3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to muscarinic acetylcholine receptor M4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to muscarinic acetylcholine receptor M5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to SERT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to NET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to MOR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to DOR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to KOR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1B receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1D receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT1E receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT5A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT6 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT7 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to 5HT7A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50539742(CHEMBL4642292)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to sigma2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303985(CHEMBL567269 | Ethyl 2,2-Dimethyl-3-(4-(2-(4-methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303984(CHEMBL565379 | Ethyl 2-Methyl-2-(4-((4-methyl-2-pr...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303983(CHEMBL565793 | ethyl 2-(4-((4-methyl-2-propyl-1H-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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