Affinity DataKi: 0.00520nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.0160nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 3.40nM ΔG°: -49.1kJ/mole IC50: 5.5nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 3.5nM ΔG°: -49.1kJ/mole IC50: 5.70nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 3.90nM ΔG°: -48.8kJ/mole IC50: 6.30nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 4.70nM ΔG°: -48.3kJ/molepH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.30nM ΔG°: -48.0kJ/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 11nM ΔG°: -46.2kJ/mole IC50: 18nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 19nM ΔG°: -44.8kJ/moleT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 35nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 48nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University Of California San Diego
University Of California San Diego
Affinity DataKi: 56nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity of compound towards Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 69nM ΔG°: -41.6kJ/mole IC50: 95nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
Affinity DataKi: 80nM ΔG°: -41.2kJ/mole IC50: 111nMpH: 7.5 T: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibitory activity against human Tryptase beta 2 expressed in yeast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair