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Found 38 with Last Name = 'karamyan' and Initial = 'vt'
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303975(3'-(4-(2-(1H-Tetrazol-5-yl)ethyl)benzyl)-1,7'-dime...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303976(3'-(2-(4-(2-(1H-Tetrazol-5-yl)ethyl)phenoxy)ethyl)...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303977(3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'-biben...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303979(CHEMBL571763 | Ethyl 3-(4-(2-(1,7'-Dimethyl-2'-pro...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303978(1-(4-(2-(1H-tetrazol-5-yl)ethyl)benzyl)-4-methyl-2...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303980(1-(4-((1H-Tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataKi:  5.06E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303984(CHEMBL565379 | Ethyl 2-Methyl-2-(4-((4-methyl-2-pr...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303985(CHEMBL567269 | Ethyl 2,2-Dimethyl-3-(4-(2-(4-methy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303986(CHEMBL584704 | Ethyl 2-Methyl-3-(4-(2-(4-methyl-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303982(CHEMBL567689 | Methyl 3-(4-((4-Methyl-2-propyl-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303983(CHEMBL565793 | ethyl 2-(4-((4-methyl-2-propyl-1H-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303981(CHEMBL567063 | Ethyl 3-(4-((4-Methyl-2-propyl-1H-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593594(CHEMBL5189177)
Affinity DataEC50:  2.48E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593595(CHEMBL5182533)
Affinity DataEC50:  3.09E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593596(CHEMBL5169334)
Affinity DataEC50:  1.36E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593597(CHEMBL5173246)
Affinity DataEC50:  3.61E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593598(CHEMBL5188276)
Affinity DataEC50:  2.86E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593599(CHEMBL5200789)
Affinity DataEC50:  2.28E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593600(CHEMBL5201458)
Affinity DataEC50:  3.22E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593601(CHEMBL5195334)
Affinity DataEC50:  1.56E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593602(CHEMBL5207768)
Affinity DataEC50:  9.06E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593603(CHEMBL5193388)
Affinity DataEC50:  2.67E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593604(CHEMBL5208268)
Affinity DataEC50:  2.79E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593593(CHEMBL5199687)
Affinity DataEC50:  7.82E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593592(CHEMBL5178128)
Affinity DataEC50:  3.75E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593591(CHEMBL5181289)
Affinity DataEC50:  1.17E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593590(CHEMBL5173065)
Affinity DataEC50:  5.21E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593589(CHEMBL5198439)
Affinity DataEC50:  2.14E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593588(CHEMBL5201850)
Affinity DataEC50:  2.41E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593587(CHEMBL5175059)
Affinity DataEC50:  1.21E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593586(CHEMBL5189262)
Affinity DataEC50:  1.05E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593585(CHEMBL5180986)
Affinity DataEC50:  5.35E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593584(CHEMBL5174943)
Affinity DataEC50:  4.51E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593583(CHEMBL5179858)
Affinity DataEC50:  1.14E+5nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeurolysin, mitochondrial(Rattus norvegicus)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50593605(CHEMBL5172435)
Affinity DataEC50:  2.52E+4nMAssay Description:Activation of recombinant rat Nln using MCA-Pro-Leu-Gly-Pro-D-Lys (DNP)-OH as substrate preincubated for 10 mins followed by substrate addition and m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50303986(CHEMBL584704 | Ethyl 2-Methyl-3-(4-(2-(4-methyl-2-...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at PPARalpha assessed as receptor transactivation by reporter gene assayMore data for this Ligand-Target Pair