TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 0.745nMAssay Description:Displacement of [3H]-N6-PIA binding from A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 0.745nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 0.939nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 1.08nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 1.56nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 2.73nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 6.81nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 7.55nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 15.7nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 35.3nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 37.2nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
Affinity DataKi: 44.5nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 56.3nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 88.3nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:Affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:Inhibition of factor 7a (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Binding affinity towards Adenosine A2a receptor by inhibition of [3H]-CGS-21,680 binding to rat brain striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 247nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 256nMAssay Description:Displacement of [3H]-N6-PIA from Adenosine A1 receptor from rat whole brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 428nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 452nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibition of thrombin (unknown origin) by spectrophotometric assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 551nMAssay Description:Binding affinity for Adenosine A1 receptor by inhibition of [3H]-PIA binding to whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 553nMAssay Description:Affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 610nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 644nMAssay Description:Affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 648nMAssay Description:Displacement of [3H]-CGS-21,680 (Kd, 14.9 nM) from A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 796nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Displacement of [3H]-CGS-21,680 (Kd, 14.9 nM) from A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair