Affinity DataKd: 10nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 23nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 39nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 55nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 102nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 209nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 209nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 358nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.09E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.38E+3nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.78E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.78E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.88E+3nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 1.88E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 3.94E+3nMAssay Description:Displacement of [3H]S-glutamate from rat GluR5 S1S2 ligand binding core expressed in Escherichia coli (DE3)More data for this Ligand-Target Pair
Affinity DataKd: 4.68E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.80E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.94E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 8.17E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 9.25E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 9.25E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.05E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 4.91E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.37E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 6.02E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 6.05E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 7.31E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 7.31E+4nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKi: 0.0810nMAssay Description:Displacement of [3H]SYM 2081 from rat recombinant GluR5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.663nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR5More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK1 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 1.11nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR5More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Yokohama City University
Curated by ChEMBL
Yokohama City University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK2 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]SYM 2081 from rat recombinant GluR5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair