Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50013264
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  390nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128313(CHEMBL57543 | N-[1-(3,5-Dimethyl-benzoyl)-cyclopen...)
Affinity DataEC50:  1.91E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128299(4-Methyl-benzo[1,3]dioxole-5-carboxylic acid [1-(3...)
Affinity DataEC50:  3.68E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128300(CHEMBL55869 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.41E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(CHEMBL54575 | N-[1-(3,5-Dimethyl-benzoyl)-cyclobut...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(CHEMBL54575 | N-[1-(3,5-Dimethyl-benzoyl)-cyclobut...)
Affinity DataEC50:  8.52E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(CHEMBL59044 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.81E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128303(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclopentyl]-2-...)
Affinity DataEC50:  6.61E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128304(CHEMBL52252 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.80E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  280nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  100nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128306(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cycloheptyl]-2-...)
Affinity DataEC50:  1.94E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  740nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(CHEMBL59044 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.25E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128307(CHEMBL56411 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(CHEMBL299671 | N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl...)
Affinity DataEC50:  4.53E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128307(CHEMBL56411 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128308(CHEMBL293929 | N-[4-(3,5-Dimethyl-benzoyl)-1,1-dio...)
Affinity DataEC50:  1.50E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128306(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cycloheptyl]-2-...)
Affinity DataEC50:  3.36E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128309(3,5-Dimethyl-benzoic acid N-tert-butyl-N'-(2-ethyl...)
Affinity DataEC50:  250nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128310(CHEMBL55953 | N-[1-(3,5-Dimethyl-benzoyl)-cyclopro...)
Affinity DataEC50:  2.04E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128303(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclopentyl]-2-...)
Affinity DataEC50:  5.16E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128300(CHEMBL55869 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.11E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128312(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclohexyl]-2-m...)
Affinity DataEC50:  980nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128311(CHEMBL54983 | N-[2-(3,5-Dimethyl-phenyl)-1,1-dimet...)
Affinity DataEC50:  4.20E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128312(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclohexyl]-2-m...)
Affinity DataEC50:  1.03E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128310(CHEMBL55953 | N-[1-(3,5-Dimethyl-benzoyl)-cyclopro...)
Affinity DataEC50:  3.33E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128304(CHEMBL52252 | N-[4-(3,5-Dimethyl-benzoyl)-tetrahyd...)
Affinity DataEC50:  1.60E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128309(3,5-Dimethyl-benzoic acid N-tert-butyl-N'-(2-ethyl...)
Affinity DataEC50:  410nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128313(CHEMBL57543 | N-[1-(3,5-Dimethyl-benzoyl)-cyclopen...)
Affinity DataEC50:  1.87E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(CHEMBL55108 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohex...)
Affinity DataEC50:  1.51E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128308(CHEMBL293929 | N-[4-(3,5-Dimethyl-benzoyl)-1,1-dio...)
Affinity DataEC50:  3.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128311(CHEMBL54983 | N-[2-(3,5-Dimethyl-phenyl)-1,1-dimet...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128315(CHEMBL300989 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohe...)
Affinity DataEC50:  1.61E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128315(CHEMBL300989 | N-[1-(3,5-Dimethyl-benzoyl)-cyclohe...)
Affinity DataEC50:  2.97E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128299(4-Methyl-benzo[1,3]dioxole-5-carboxylic acid [1-(3...)
Affinity DataEC50:  3.22E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(CHEMBL299671 | N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl...)
Affinity DataEC50:  6.23E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed