Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Ecdysone receptor' and Ligand = 'BDBM50128305'
TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  280nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  100nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed