BDBM50128305 3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenzoyl)-2-(1,1-dimethylethyl)hydrazide::CHEMBL55772::N'-(tert-butyl)-N'-(3,5-dimethylbenzoyl)-3-methoxy-2-methylbenzohydrazide::N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2-methylbenzohydrazide::N-tert-butyl-N'-(3-methoxy-o-toluoyl)-3,5-xylohydrazide::methoxyfenozide

SMILES COc1cccc(C(=O)NN(C(=O)c2cc(C)cc(C)c2)C(C)(C)C)c1C

InChI Key InChIKey=QCAWEPFNJXQPAN-UHFFFAOYSA-N

Data  1 IC50  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50128305   

TargetEcdysone receptor(Choristoneura fumiferana)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  280nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  100nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataIC50:  4.43E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ultraspiracle(Drosophila melanogaster)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Bombyx mori)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor(Spodoptera littoralis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed