Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- Acid-sensing ion channel 1
- Adenosine A1 receptor
- Adenosine Receptors A2a (A2a)
- Adenosine receptor A1
- Adenosine receptor A2a
- Adrenaline alpha1
- Adrenaline alpha2
- Adrenergic Alpha
- Alpha-1A adrenergic receptor
- Amiloride-sensitive cation channel 3
- Amiloride-sensitive sodium channel alpha-subunit
- Beta-1 adrenergic receptor
- Bile salt export pump
- CCKBR
- Calcium channel (DHP)
- Calcium release-activated calcium channel
- Coagulation factor X
- Coagulation factor XI
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(2) dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- Glycine
- HTR1D
- HTR2C
- Histamine H1 receptor
- Kappa-type opioid receptor
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Opioid receptors; mu & delta
- Plasma kallikrein
- Plasminogen
- Prothrombin
- Serine/threonine-protein kinase D1
- Serine/threonine-protein kinase PLK1
- Serotonin 1B/1D receptor
- Sodium channel protein type 5 subunit alpha
- Sodium/hydrogen exchanger
- Sodium/hydrogen exchanger 1
- Substance K
- TRH
- Tissue-type plasminogen activator
- Trypsin
- Urokinase-type plasminogen activator
- Urokinase-type plasminogen activator (uPA)
- Urokinase-type plasminogen activator/surface receptor
- Vascular adhesion protein 1 (VAP-1)
- Vitamin K-dependent protein C
- adrenergic Alpha2
- 3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinamide;hydrochloride
- 3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-carboxamide
- Amiloride
- Amipramidin
- CHEMBL945
- 3-phosphoinositide dependent protein kinase-1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1
- ALK tyrosine kinase receptor
- Angiopoietin-1 receptor
- Aurora kinase A/Targeting protein for Xklp2
- B-RAF V600E
- CAMK2A
- Casein kinase I isoform delta
- Cyclin-dependent kinase 2
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Ephrin type-A receptor 1 (EPHA1)
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 1
- Hepatocyte growth factor receptor
- Inhibitor of nuclear factor kappa-B kinase subunit beta
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- MAP kinase-activated protein kinase 2
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 9
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Platelet-derived growth factor receptor beta
- Protein kinase C alpha type
- Proto-oncogene tyrosine-protein kinase Src
- RAC-alpha serine/threonine-protein kinase
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase (P70S6K)
- Ribosomal protein S6 kinase alpha 5
- Ribosomal protein S6 kinase alpha-3
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase D1
- Serine/threonine-protein kinase MARK1
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek2
- Serine/threonine-protein kinase Sgk1
- Serine/threonine-protein kinase TAO2
- Serine/threonine-protein kinase pim-1
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase Fes/Fps
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor UFO
- Vascular endothelial growth factor receptor 2
- cAMP-dependent protein kinase (PKA)
- p21-Activated kinase 2 (PAK2)
55 IC50
- US9365572, 5
- 5-HT1
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- ADRA1A
- ADRA1B
- ADRA2C
- Adenosine receptor A1
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- Calcium channel
- Calcium channel (Type L)
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- DRD1
- DRD2
- Dopamine receptor
- GABA receptor gamma-1 subunit
- GST-MALT lymphoma-associated translocation (MALT1)
- HTR6
- Histamine H1 receptor
- Muscarinic acetylcholine receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Pleiotropic ABC efflux transporter of multiple drugs
- Potassium voltage-gated channel subfamily H member 2
- Proteasome subunit alpha type-6
- Replicase polyprotein 1ab
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- Sigma non-opioid intracellular receptor 1
- Sodium channel protein type 5 subunit alpha
- Sodium channel protein type I I alpha subunit
- Voltage-dependent L-type calcium channel subunit alpha-1C
- Voltage-gated L-type calcium channel
- adrenergic Alpha2
- (Thioridazine)10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine
- 10-(2-(1-methylpiperidin-2-yl)ethyl)-2-(methylthio)-10H-phenothiazine
- 10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine
- 10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsulfanyl-10H-phenothiazine (thioridazine)
- CHEMBL479
- MELLARIL
- MELLARIL-S
- THIORIDAZINE
- TP-21
- US9504692, Thioridazine
- Aurora kinase A/Targeting protein for Xklp2
- Aurora kinase B
- Axin-1/Glycogen synthase kinase-3 beta
- BDNF/NT-3 growth factors receptor
- Casein kinase I isoform delta
- Cyclin-dependent kinase 1
- Cyclin-dependent-like kinase 5
- Death-associated protein kinase 3
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Ephrin type-A receptor 2
- Epidermal growth factor receptor
- Glycogen synthase kinase-3
- High affinity nerve growth factor receptor
- Insulin receptor
- Insulin-like growth factor I receptor
- MAP kinase-activated protein kinase 3
- Macrophage colony-stimulating factor 1 receptor (CSF1R)
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 12
- Mitogen-activated protein kinase 13 (MAPK13)
- Non-receptor tyrosine-protein kinase TYK2
- PAK 1/CDC42
- Protein kinase C delta type
- Protein kinase C, eta
- Protein kinase C, gamma
- Proto-oncogene tyrosine-protein kinase Src
- Receptor protein-tyrosine kinase erbB-4
- Receptor tyrosine-protein kinase erbB-2
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Serine/threonine-protein kinase AKT
- Serine/threonine-protein kinase AKT2
- Serine/threonine-protein kinase CHK2
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase D2
- Serine/threonine-protein kinase MRCK alpha
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek2
- Serine/threonine-protein kinase PAK 4
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK3
- Serine/threonine-protein kinase Sgk1
- Serine/threonine-protein kinase pim-1
- Serine/threonine-protein kinase pim-2
- Tyrosine-protein kinase Blk
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Vascular endothelial growth factor receptor 2
- Vascular endothelial growth factor receptor 3
56 IC50
- CHEMBL1090360
- N-(3-(5-(2-(3-morpholinophenylamino)pyrimidin-4-yl)imidazo[2,1-b]thiazol-6-yl)phenyl)-2-phenylacetamide
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 4 (5-HT4)
- 5-hydroxytryptamine receptor 7
- Acetylcholinesterase
- Adenosine receptor A1
- Adenosine receptor A2a
- Adenosine receptor A3
- Adrenergic alpha1B
- Alpha-1A adrenergic receptor
- Alpha-1D adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Amine oxidase (flavin-containing) A
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Cannabinoid receptor 1
- Cholecystokinin receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Dopamine receptor D2L/neurotensin receptor NTS1
- Endothelin-1 receptor
- Glucocorticoid receptor
- High-affinity choline transporter
- Histamine H1 receptor
- Histamine H2 receptor
- Histamine H3 receptor
- Imidazoline receptor 1 (I1R)
- Kappa-type opioid receptor
- Melanin-concentrating hormone receptor
- Melanocortin receptor 4
- Melatonin receptor
- Mitogen-activated protein kinase 14
- Mu-type opioid receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- Neurokinin 1 receptor
- Neurokinin 2 receptor
- Neuronal acetylcholine receptor Alpha-4/Beta-2
- Neuropeptide Y receptor type 1
- Potassium voltage-gated channel subfamily H member 2
- Ribosyldihydronicotinamide dehydrogenase [quinone]
- Sodium-dependent dopamine transporter
- Sodium-dependent noradrenaline transporter
- Sodium-dependent serotonin transporter
- Tyrosine-protein kinase Lyn
- CHEMBL1242923
- N-{1-[3-(3-Oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]-piperidin-4-yl}-2-phenylacetamide
- 5-HT3A Serotonin Receptor
- 5-HT5B
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 3A
- Adrenergic Alpha
- Adrenergic receptor beta
- Alpha-2A adrenergic receptor
- Bile salt export pump
- CCKBR
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cholecystokinin receptor
- Cytochrome P450 3A
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Glycine receptor alpha-4 chain
- HTR1D
- HTR3A
- HTR4
- Histamine H1 receptor
- Histamine H3 receptor
- Imidazoline receptor 1 (I1R)
- Interleukin-6 receptor alpha chain
- Kappa-type opioid receptor
- Leukotriene B4
- Mu-type opioid receptor
- Multidrug and toxin extrusion protein 1
- Multidrug and toxin extrusion protein 2
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- NMDA receptor subunit 2C (GluN2C)
- Neuronal acetylcholine receptor
- Neuronal acetylcholine receptor Alpha-4/Beta-2
- Neuronal acetylcholine receptor protein alpha-7 subunit
- Neuronal acetylcholine receptor; alpha3/beta4
- Opioid receptors; mu & delta
- Potassium voltage-gated channel subfamily H member 2
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin 3 receptor (5HT3)
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- Sodium-dependent serotonin transporter
- Solute carrier family 22 member 2
- Solute carrier family 22 member 3
- Thyrotropin-releasing hormone receptor
- Voltage-gated L-type calcium channel
- CAS_68647
- NSC_68647
- ONDANSETRON
- Ondansetron hydrochloride