Search by Compound Name
Compounds Sorted by Binding Targets per Compound
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 2930 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 73 74 75 76 77 79 81 84 86 89 95
96 100 108 109 120 124 130 137 143 154 156 168 186 224 240 259 276 278 284 303
304 310 315 323 339 369 370 371 372 373 374 375 376 377 378 380 381 383 384
385 386 388 389 390 391 392 393 394 395 397 398 401 403 404 406 408 418 427
429 443 447 515
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
- 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2B
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 6
- 5-hydroxytryptamine receptor 7
- 5-hydroxytryptamine receptor 7 (5HT7)
- Adrenergic receptor alpha-1
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor
- Bile salt export pump
- CCKBR
- Calcium channel
- Canalicular multispecific organic anion transporter 1
- Canalicular multispecific organic anion transporter 2
- Cholecystokinin B
- Cholinergic, muscarinic
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(1B) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- D(4) dopamine receptor
- Delta-type opioid receptor
- Dihydrofolate Reductase (DHFR)
- Dopamine receptor
- Gamma-aminobutyric acid receptor subunit alpha-1
- HTR1D
- HTR2C
- HTR6
- Histamine H1 receptor
- Histone H1
- Kappa-type opioid receptor
- Mu-type opioid receptor
- Multidrug resistance-associated protein 4
- Muscarinic acetylcholine receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M2 and M4
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- Muscarinic acetylcholine receptor M5
- NT
- Norepinephrine transporter
- Potassium voltage-gated channel subfamily H member 2
- Prostanoid TP receptor
- Serotonin (5-HT) receptor
- Serotonin 1B/1D receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Sigma non-opioid intracellular receptor 1
- Sodium channel protein type 5 subunit alpha
- Sodium-dependent dopamine transporter
- Sodium-dependent serotonin transporter
- Substance P
- Transporter
- Voltage-dependent L-type calcium channel subunit alpha-1C
- Voltage-gated sodium channel subunit alpha Nav1.8
- adrenergic Alpha2
- 2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol
- 2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-1-yl)ethoxy]ethanol
- CHEMBL716
- QUETIAPINE
- Angiopoietin-1 receptor
- Aurora kinase A/Targeting protein for Xklp2
- Axin-1/Glycogen synthase kinase-3 beta
- CaM kinase I delta
- CaM kinase IV
- Ceramide kinase
- Cyclin-dependent kinase 1
- Cytoplasmic tyrosine-protein kinase BMX
- Death-associated protein kinase 3
- Dual specificity mitogen-activated protein kinase kinase 1
- Dual specificity mitogen-activated protein kinase kinase 6
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Ephrin type-B receptor 2
- Epidermal growth factor receptor
- Fibroblast growth factor receptor 4
- Focal adhesion kinase 1
- Indoleamine 2,3-dioxygenase
- Inhibitor of nuclear factor kappa-B kinase subunit alpha
- Insulin receptor
- Insulin-like growth factor I receptor
- Interleukin-1 receptor-associated kinase 4
- MAP kinase-activated protein kinase 5
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 11
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 3
- Mitogen-activated protein kinase 8
- Mitogen-activated protein kinase kinase kinase 7
- Mitogen-activated protein kinase kinase kinase 8
- PKC alpha and beta-2
- Platelet-derived growth factor receptor alpha
- Protein kinase C theta type
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- RAC-alpha serine/threonine-protein kinase
- RAF proto-oncogene serine/threonine-protein kinase
- Receptor protein-tyrosine kinase erbB-4
- Rho-associated protein kinase 2
- Ribosomal protein S6 kinase (P70S6K)
- Ribosomal protein S6 kinase alpha 1
- Ribosomal protein S6 kinase alpha 5
- Serine/threonine-protein kinase Chk1/2
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase Nek1
- Serine/threonine-protein kinase PLK3
- Serine/threonine-protein kinase Sgk1
- Serine/threonine-protein kinase TBK1
- Serine/threonine-protein kinase pim-1
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase FER
- Tyrosine-protein kinase Fes/Fps
- Tyrosine-protein kinase Fyn
- Tyrosine-protein kinase HCK
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase Yes
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor FLT3
- Vascular endothelial growth factor receptor 2
73 Ki
- (S)-3-(4-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)benzoylamino)-5-(6-(methylamino)pyrazin-2-yl)-(1H)-pyridin-2-one
- CHEMBL1765781