BDBM185344 US9156830, I-50

SMILES OCCc1nnc(o1)-c1cnc(C2=CCN(CC2)C(=O)Nc2ccc(c(Cl)c2)C(F)(F)F)c(Cl)c1

InChI Key InChIKey=KLOWQQXEIZVHIP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 185344   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM185344(US9156830, I-50)
Affinity DataIC50:  60.8nMpH: 7.4Assay Description:Two days prior to performing this assay, cells are seeded on poly-D-lysine-coated 96-well clear-bottom black plates (commercially available from Bect...More data for this Ligand-Target Pair
In DepthDetails US Patent