BDBM50056412 4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolidin-1-yl-ethyl ester::CHEMBL156970
SMILES COc1cc(N)c(Cl)cc1C(=O)OCCN1CCCC1
InChI Key InChIKey=XEZGQZRJNWWNJR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50056412
Affinity DataKi: 5.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair