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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50056412'
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056412(4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolid...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056412(4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolid...)
Affinity DataIC50:  200nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50056412(4-Amino-5-chloro-2-methoxy-benzoic acid 2-pyrrolid...)
Affinity DataEC50:  40nMAssay Description:5-hydroxytryptamine 4 receptor agonist activity, concentration which gave 50% increase in the response to electrically-stimulated myenteric plexus an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed