BDBM50322249 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)-methyl)piperidin-4-ol oxalate::CHEMBL1173366
SMILES OC1(CCN(Cc2c[nH]c3ccc(OCCF)cc23)CC1)c1ccc(Br)cc1
InChI Key InChIKey=VGEYSHNQKQOFLR-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50322249
Affinity DataKi: 13.8nMAssay Description:Displacement of [125I]ABN from human dopamine D2 long receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Displacement of [125I]ABN from human dopamine D3 receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 227nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain homogenates after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 344nMAssay Description:Displacement of [125I]ABN from human dopamine D4 receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair