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Found 336 with Last Name = 'gioiello' and Initial = 'a'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50022802(CHEMBL2046866)
Affinity DataKi:  3.30nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50022803(CHEMBL5288617)
Affinity DataKi:  5.10nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50429537(CHEMBL2333770)
Affinity DataKi:  6nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM129261(US8815951, 297)
Affinity DataKi:  7nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50120392(CHEMBL5282574)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50056299(CHEMBL5288434)
Affinity DataKi:  99nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50541371(CHEMBL4641964)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of alpha1B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50541370(CHEMBL2146625)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of alpha1B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50187004(3-(3,4-dioxo-2-(phenylamino)cyclobut-1-enylamino)-...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50200880((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-...)
Affinity DataIC50:  2.60nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50432620(CHEMBL2347192)
Affinity DataIC50:  12nMAssay Description:Inhibition of BACE1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataIC50:  15nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
The University of Georgia

Curated by ChEMBL
LigandPNGBDBM50200880((R)-2-hydroxy-N,N-dimethyl-3-(2-(1-(5-methylfuran-...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataIC50:  60nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046166(CHEMBL3310984)
Affinity DataIC50:  70nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataIC50:  73nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046169(CHEMBL3310985)
Affinity DataIC50:  74nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046167(CHEMBL1332361)
Affinity DataIC50:  76nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046170(CHEMBL1533910)
Affinity DataIC50:  79nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM46912(4-methyl-N-(2-phenylphenyl)benzenesulfonamide | ML...)
Affinity DataIC50:  90nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataIC50:  90nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046168(CHEMBL1372946)
Affinity DataIC50:  93nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046165(CHEMBL1621411)
Affinity DataIC50:  94nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046171(CHEMBL362436)
Affinity DataIC50:  128nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046171(CHEMBL362436)
Affinity DataIC50:  174nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046170(CHEMBL1533910)
Affinity DataIC50:  179nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50016567((Toluene-4-sulfonylamino)-acetic acid | CHEMBL2874...)
Affinity DataIC50:  217nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Regina Elena National Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50260175(CHEMBL4088384)
Affinity DataIC50:  223nMAssay Description:Displacement of [3H]R-1881 from Androgen receptor of PC3-AR cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM46912(4-methyl-N-(2-phenylphenyl)benzenesulfonamide | ML...)
Affinity DataIC50:  226nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046166(CHEMBL3310984)
Affinity DataIC50:  248nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046169(CHEMBL3310985)
Affinity DataIC50:  255nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046168(CHEMBL1372946)
Affinity DataIC50:  266nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataIC50:  295nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046165(CHEMBL1621411)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50016567((Toluene-4-sulfonylamino)-acetic acid | CHEMBL2874...)
Affinity DataIC50:  3.62E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046167(CHEMBL1332361)
Affinity DataIC50:  4.28E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM46912(4-methyl-N-(2-phenylphenyl)benzenesulfonamide | ML...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046165(CHEMBL1621411)
Affinity DataIC50:  6.67E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046171(CHEMBL362436)
Affinity DataIC50:  7.32E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046166(CHEMBL3310984)
Affinity DataIC50:  8.07E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataIC50:  8.44E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 12(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50016567((Toluene-4-sulfonylamino)-acetic acid | CHEMBL2874...)
Affinity DataIC50:  8.57E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM46912(4-methyl-N-(2-phenylphenyl)benzenesulfonamide | ML...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046170(CHEMBL1533910)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046167(CHEMBL1332361)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046169(CHEMBL3310985)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046168(CHEMBL1372946)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50046165(CHEMBL1621411)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM50428400(CA inhibitor, 2 | CHEMBL182659 | [(4-Methylphenyl)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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