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Found 187 with Last Name = 'baumgold' and Initial = 'j'
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.5nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.70nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  1.80nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.90nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataKi:  2.10nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine rec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280621(4-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-3...)
Affinity DataKi:  2.40nMAssay Description:Inhibitory constant of the compound was determined by the inhibition of [3H]-N-methylscopolamine (NMS) binding to m1 receptor of transfected A9L cell...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005684(2-Cyclohexyl-2-phenyl-propionic acid 3-diethylamin...)
Affinity DataKi:  2.90nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012344(11-{2-[4-(10-Diethylamino-decyl)-piperazin-1-yl]-a...)
Affinity DataKi:  3nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012336(11-(2-{4-[10-(2-Methoxy-benzylamino)-decyl]-pipera...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50280621(4-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-3...)
Affinity DataKi:  3.70nMAssay Description:Inhibitory constant of the compound was determined by the inhibition of [3H]-N-methylscopolamine (NMS) binding to Muscarinic acetylcholine receptor M...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005684(2-Cyclohexyl-2-phenyl-propionic acid 3-diethylamin...)
Affinity DataKi:  4nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005686(2-Cyclohexyl-2-phenyl-propionic acid 2-diethylamin...)
Affinity DataKi:  4nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005684(2-Cyclohexyl-2-phenyl-propionic acid 3-diethylamin...)
Affinity DataKi:  4.60nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  6.90nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataKi:  7.40nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataKi:  7.70nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine rec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataKi:  9.30nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine rec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005686(2-Cyclohexyl-2-phenyl-propionic acid 2-diethylamin...)
Affinity DataKi:  9.90nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Muscarinic acetylcholine receptor M...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012353(11-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  12nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012344(11-{2-[4-(10-Diethylamino-decyl)-piperazin-1-yl]-a...)
Affinity DataKi:  14nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012353(11-{2-[4-(10-Amino-decyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  16nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  17nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012348(2-(6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  18nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012348(2-(6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  18nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005686(2-Cyclohexyl-2-phenyl-propionic acid 2-diethylamin...)
Affinity DataKi:  19nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012360(11-{2-[4-(8-Amino-octyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  20nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005684(2-Cyclohexyl-2-phenyl-propionic acid 3-diethylamin...)
Affinity DataKi:  20nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012357(2-(5-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  20nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  21nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012336(11-(2-{4-[10-(2-Methoxy-benzylamino)-decyl]-pipera...)
Affinity DataKi:  22nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005686(2-Cyclohexyl-2-phenyl-propionic acid 2-diethylamin...)
Affinity DataKi:  23nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  23nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to muscarinic acetylcholine receptor M4 of rat heart NG108-15 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012345(11-{2-[4-(9-Amino-nonyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  24nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012345(11-{2-[4-(9-Amino-nonyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  24nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012360(11-{2-[4-(8-Amino-octyl)-piperazin-1-yl]-acetyl}-5...)
Affinity DataKi:  26nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  27nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  29nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005682(2-Cyclohexyl-2-phenyl-propionic acid 4-dimethylami...)
Affinity DataKi:  31nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  37nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005682(2-Cyclohexyl-2-phenyl-propionic acid 4-dimethylami...)
Affinity DataKi:  41nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012371(CHEMBL70154 | N-(10-{4-[2-Oxo-2-(6-oxo-5,6-dihydro...)
Affinity DataKi:  43nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012338((6-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido[3...)
Affinity DataKi:  46nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M3 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  50nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M2 of rat heart tissue membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012327(CHEMBL68292 | N-(9-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  50nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012365(11-{2-[4-(2-Chloro-ethyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  52nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012327(CHEMBL68292 | N-(9-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-...)
Affinity DataKi:  52nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012351(11-{2-[4-(7-Amino-heptyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  57nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M2 of rat heart tissue membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012357(2-(5-{4-[2-Oxo-2-(6-oxo-5,6-dihydro-benzo[e]pyrido...)
Affinity DataKi:  60nMAssay Description:Inhibition of binding of [3H]-N-methylscopolamine to muscarinic acetylcholine receptor M1 of transfected rat A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005682(2-Cyclohexyl-2-phenyl-propionic acid 4-dimethylami...)
Affinity DataKi:  66nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50012351(11-{2-[4-(7-Amino-heptyl)-piperazin-1-yl]-acetyl}-...)
Affinity DataKi:  66nMAssay Description:Inhibition of binding of [3H]-N-Methyl-scopolamine to Muscarinic acetylcholine receptor M1 of transfected A9L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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