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Found 30 with Last Name = 'chekanov' and Initial = 'mo'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM32315(CHEMBL1345690 | MLS000715851 | SMR000277368 | cid_...)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human ASK1 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248081(3-{[2-chloro-4-(1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248071(3-{[4-(1,1-dioxido-3-oxoisothiazolidin-2-yl)benzoy...)
Affinity DataIC50:  1.80E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248083(4-{[2-chloro-4-(1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50:  3.00E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM32315(CHEMBL1345690 | MLS000715851 | SMR000277368 | cid_...)
Affinity DataIC50:  3.00E+3nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248074(3-{[4-(4-methyl-1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50:  3.10E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248088(4-{[2-chloro-4-(4-methyl-1,1-dioxido-3-oxoisothiaz...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248085(3-{[2-chloro-4-(4-methyl-1,1-dioxido-3-oxoisothiaz...)
Affinity DataIC50:  3.60E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248087(3-{[2-chloro-4-(4-methyl-1,1-dioxido-3-oxoisothiaz...)
Affinity DataIC50:  3.70E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342272(3-Methyl-1-(methylamino)-3H-naphtho[1,2,3-de]quino...)
Affinity DataIC50:  4.70E+3nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248086(5-{[2-chloro-4-(4-methyl-1,1-dioxido-3-oxoisothiaz...)
Affinity DataIC50:  6.00E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248078(3-{[4-(4,4-dimethyl-1,1-dioxido-3-oxoisothiazolidi...)
Affinity DataIC50:  8.00E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248072(5-{[4-(1,1-dioxido-3-oxoisothiazolidin-2-yl)benzoy...)
Affinity DataIC50:  8.00E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248082(5-{[2-chloro-4-(1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM39880(1-(ethylamino)-3-methyl-3H-naphtho[1,2,3-de]quinol...)
Affinity DataIC50:  1.00E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248073(4-{[4-(1,1-dioxido-3-oxoisothiazolidin-2-yl)benzoy...)
Affinity DataIC50:  1.40E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342273(1-Acetyl-3H-naphtho[1,2,3-de]quinoline-2,7-dione |...)
Affinity DataIC50:  1.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248076(4-hydroxy-3-{[4-(4-methyl-1,1-dioxido-3-oxoisothia...)
Affinity DataIC50:  1.60E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248077(2-hydroxy-4-{[4-(4-methyl-1,1-dioxido-3-oxoisothia...)
Affinity DataIC50:  1.95E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM32006(1-(2-Hydroxy-ethylamino)-3-methyl-3H-naphtho[1,2,3...)
Affinity DataIC50:  2.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248075(2-hydroxy-5-{[4-(4-methyl-1,1-dioxido-3-oxoisothia...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248092(4-{[4-(4-methyl-1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248091(N-[4-(4-methyl-1,1-dioxido-3-oxoisothiazolidin-2-y...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248090(N-[4-(4-methyl-1,1-dioxido-3-oxoisothiazolidin-2-y...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248089(Methyl 5-{[2-chloro-4-(4-methyl-1,1-dioxido-3-oxoi...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248079(5-{[4-(4,4-dimethyl-1,1-dioxido-3-oxoisothiazolidi...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248084(4-{[2-chloro-4-(1,1-dioxido-3-oxoisothiazolidin-2-...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Nas of Ukraine

LigandPNGBDBM248080(4-{[4-(4,4-dimethyl-1,1-dioxido-3-oxoisothiazolidi...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Each test was performed twice in a total reaction volume of 30 μL, containing 6 μg of peptide substrate RRRDDDSDDD (New England Biolabs (UK) Lt...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342274(1-Benzoyl-3-methyl-3H-naphtho[1,2,3-de]quinoline-2...)
Affinity DataIC50:  3.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Nas Of Ukraine

Curated by ChEMBL
LigandPNGBDBM50342275(1-Acetyl-4-methyl-3H-naphtho[1,2,3-de]quinoline-2,...)
Affinity DataIC50:  3.50E+4nMAssay Description:Competitive inhibition of human ASK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed