Compile Data Set for Download or QSAR
maximum 50k data
Found 215 with Last Name = 'dulski' and Initial = 'p'
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50238632((6S,9S,12S,14aR)-6-((S)-sec-Butyl)-9-(1-methoxy-1H...)
Affinity DataKi:  8nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366737(CHEMBL1793971)
Affinity DataKi:  10nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366726(CHEMBL1793982)
Affinity DataKi:  20nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366733(CHEMBL1793973)
Affinity DataKi:  30nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366749(CHEMBL1793983)
Affinity DataKi:  50nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366736(CHEMBL1793972)
Affinity DataKi:  70nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366727(CHEMBL1793981)
Affinity DataKi:  100nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366729(CHEMBL1793969)
Affinity DataKi:  200nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366752(CHEMBL1793970)
Affinity DataKi:  250nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366728(CHEMBL1793978)
Affinity DataKi:  400nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366750(CHEMBL1793987)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards HDAC enzyme derived from Eimeria tenella protozoaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168170(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.0460nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374578(CHEMBL401749)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374594(CHEMBL444009)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366693(CHEMBL1793812)
Affinity DataIC50: <0.100nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) derived from partially purified extracts of human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168185(4-[2-(3-Bromo-4-fluoro-phenyl)-5-(1-methyl-piperid...)
Affinity DataIC50:  0.150nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171694((R)-5-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.160nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374591(CHEMBL255128)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374587(CHEMBL272573)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366738(CHEMBL1793985)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Cryptosporidium parvum)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366738(CHEMBL1793985)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase enzyme derived from partially purified extracts of Eimeria tenella protozoa using [3H]11 as radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366696(CHEMBL1793811)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) derived from partially purified extracts of human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50218940(CHEMBL1793991)
Affinity DataIC50:  0.200nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) enzyme derived from partially purified extracts of human HeLa cells using [3H]11 as radioligan...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168208(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374588(CHEMBL255381)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168187(4-{2-(4-Fluoro-phenyl)-5-[1-(1-methyl-azetidin-2-y...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168202(2-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374592(CHEMBL271922)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168206(4-[5-(1-Ethyl-piperidin-4-yl)-2-(4-fluoro-phenyl)-...)
Affinity DataIC50:  0.280nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366712(CHEMBL1793822)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) derived from partially purified extracts of human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168192(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.320nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374580(CHEMBL271638)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50183915((5-(4-fluorophenyl)-4-(pyridin-4-yl)-1H-pyrrol-2-y...)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374590(CHEMBL406910)
Affinity DataIC50:  0.360nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171685(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.380nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374593(CHEMBL429745)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171698(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50366713(CHEMBL1793816)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against histone deacetylase (HDAC) derived from partially purified extracts of human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171707(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.410nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168190(4-[2-(3-Chloro-4-fluoro-phenyl)-5-(1-methyl-piperi...)
Affinity DataIC50:  0.440nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171705(1-Benzyloxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-...)
Affinity DataIC50:  0.470nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171699((S)-1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-py...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171693(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168176(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.530nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168176(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.530nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171695((R)1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyr...)
Affinity DataIC50:  0.560nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171688(1-Ethoxy-3-{4-[5-(4-fluoro-phenyl)-4-pyridin-4-yl-...)
Affinity DataIC50:  0.590nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171702(1-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory activity against cGMP-dependent protein kinase from Eimeria tenellaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-dependent protein kinase(Eimeria tenella)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50374585(CHEMBL255631)
Affinity DataIC50:  0.670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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