Compile Data Set for Download or QSAR
maximum 50k data
Found 275 with Last Name = 'feher' and Initial = 'v'
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136934(3',4'-Dichloro-biphenyl-3-sulfonic acid (3-chloro-...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136916(3'-Chloro-4'-fluoro-biphenyl-3-sulfonic acid (3-ch...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136914(4'-Chloro-3'-methyl-biphenyl-3-sulfonic acid (3-ch...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136919(3',4'-Difluoro-biphenyl-3-sulfonic acid (3-chloro-...)
Affinity DataKi:  8.10nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136913(CHEMBL156794 | N-(3-Chloro-7-isobutylamino-1H-inda...)
Affinity DataKi:  10.8nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136936(3'-Trifluoromethyl-biphenyl-3-sulfonic acid (3-chl...)
Affinity DataKi:  11nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136942(4'-Chloro-biphenyl-3-sulfonic acid (3-chloro-7-iso...)
Affinity DataKi:  12.5nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136911(4'-Trifluoromethyl-biphenyl-3-sulfonic acid (3-chl...)
Affinity DataKi:  13nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136918(4'-Fluoro-3'-methyl-biphenyl-3-sulfonic acid (3-ch...)
Affinity DataKi:  14.6nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136935(3'-Methylsulfanyl-biphenyl-3-sulfonic acid (3-chlo...)
Affinity DataKi:  17nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136910(3'-Trifluoromethyl-biphenyl-3-sulfonic acid (7-iso...)
Affinity DataKi:  20nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136943(3'-(2-Hydroxy-ethyl)-biphenyl-3-sulfonic acid (3-c...)
Affinity DataKi:  25nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136922(CHEMBL346924 | N-(3-Chloro-7-isobutylamino-1H-inda...)
Affinity DataKi:  28.5nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136907(CHEMBL153876 | N-(3-Chloro-7-isobutylamino-1H-inda...)
Affinity DataKi:  36nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136940(3'-Methyl-biphenyl-3-sulfonic acid (3-chloro-7-iso...)
Affinity DataKi:  36nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136930(CHEMBL154614 | N-(3-Chloro-7-isobutylamino-1H-inda...)
Affinity DataKi:  52nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136921(Biphenyl-3-sulfonic acid (3-chloro-7-isobutylamino...)
Affinity DataKi:  94nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136938(3'-Methyl-biphenyl-3-sulfonic acid (7-isobutylamin...)
Affinity DataKi:  100nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136939(3'-Ethyl-biphenyl-3-sulfonic acid (7-isobutylamino...)
Affinity DataKi:  125nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136908(CHEMBL153820 | N-(7-Isobutylamino-3-methyl-1H-inda...)
Affinity DataKi:  191nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136905(CHEMBL157223 | N-(7-Isobutylamino-3-methyl-1H-inda...)
Affinity DataKi:  240nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136926(Biphenyl-3-sulfonic acid (7-isobutylamino-3-methyl...)
Affinity DataKi:  498nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136927(4-Chloro-N-[3-chloro-7-(cyclopropylmethyl-amino)-1...)
Affinity DataKi:  500nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136923(4-Chloro-N-(3-chloro-7-isobutylamino-1H-indazol-5-...)
Affinity DataKi:  760nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136937(5-Dimethylamino-naphthalene-1-sulfonic acid (1H-in...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136931(4-Chloro-N-[3-chloro-7-(2,2-dimethyl-propylamino)-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136928(CHEMBL153833 | N-(7-Benzylamino-3-chloro-1H-indazo...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136906(4-Chloro-N-[3-chloro-7-(3-methyl-but-2-enylamino)-...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136941(4-Chloro-N-(3-chloro-7-phenethylamino-1H-indazol-5...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136944(4-Chloro-N-(3-chloro-7-ethylamino-1H-indazol-5-yl)...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136932(5-Dimethylamino-naphthalene-1-sulfonic acid (1H-in...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136925(4-Chloro-N-(3-methyl-1H-indazol-5-yl)-benzenesulfo...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136920(4-Chloro-N-[3-chloro-7-(3-methyl-butylamino)-1H-in...)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136912(4-Chloro-N-(3-chloro-1H-indazol-5-yl)-benzenesulfo...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136909(4-Chloro-N-[3-chloro-7-(3,3-dimethyl-butylamino)-1...)
Affinity DataKi:  6.50E+3nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136917(CHEMBL345702 | N-[3-Chloro-5-(4-chloro-benzenesulf...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136929(4-Chloro-N-(1H-indazol-6-yl)-benzenesulfonamide | ...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136933(5-Dimethylamino-naphthalene-1-sulfonic acid (3-chl...)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136915(4-Chloro-N-(1H-indazol-5-yl)-benzenesulfonamide | ...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase(Escherichia coli (strain K12))
Quorex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50136924(5-Dimethylamino-naphthalene-1-sulfonic acid (3-met...)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of Escherichia coli S-adenosyl homocysteine/methylthioadenosine nucleosidase (MTA/SAH nucleosidase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50232582(CHEMBL4067710)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human FLAG-tagged PLK1 expressed in baculovirus infected sf21 cells using Biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50204291(CHEMBL3953104 | US20230295171, Example 76)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50204291(CHEMBL3953104 | US20230295171, Example 76)
Affinity DataIC50:  0.501nMAssay Description:YK protein is prepared from cDNA encoding human spleen tyrosine kinase and is expressed in insect cells using a baculovirus expression vector. The cD...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM620222(BDBM50204292 | US20230295171, Example 82)
Affinity DataIC50:  0.631nMAssay Description:YK protein is prepared from cDNA encoding human spleen tyrosine kinase and is expressed in insect cells using a baculovirus expression vector. The cD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50204296(CHEMBL3941633 | US20230295171, Example 75)
Affinity DataIC50:  0.794nMAssay Description:YK protein is prepared from cDNA encoding human spleen tyrosine kinase and is expressed in insect cells using a baculovirus expression vector. The cD...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50204296(CHEMBL3941633 | US20230295171, Example 75)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM620222(BDBM50204292 | US20230295171, Example 82)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human C-terminal 6His-tagged SYK (356 to 635 residues) expressed in Sf9 insect cells using 5-carboxyfluorescein(FAM)-EEPLYWSFPAKKK-NH2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50204293(CHEMBL3983415 | US20230295171, Example 25)
Affinity DataIC50:  1nMAssay Description:YK protein is prepared from cDNA encoding human spleen tyrosine kinase and is expressed in insect cells using a baculovirus expression vector. The cD...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM50435723(CHEMBL2392549)
Affinity DataIC50:  1nMAssay Description:Inhibition of PLK1 (unknown origin) using biotin-AGAGTVPESIHSFIGDGLV as substrate by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Takeda California

Curated by ChEMBL
LigandPNGBDBM620245(US20230295171, Example 105)
Affinity DataIC50:  1nMAssay Description:YK protein is prepared from cDNA encoding human spleen tyrosine kinase and is expressed in insect cells using a baculovirus expression vector. The cD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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