TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataIC50: <300nMAssay Description:Inhibition of [3H]-dofetilide binding to human ERG expressed in HEK293 cell membranes after 1 hr by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human ERG expressed in HEK293 cells at -80 holding potential by whole patch clamp assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 4.46E+3nMAssay Description:Agonist activity at human PPARalpha receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 3.69E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 6.34E+3nMAssay Description:Agonist activity at human PPARgamma receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 1.36E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 1.17E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 2.81E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 2.55E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 4.88E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 2.97E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 2.61E+3nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nagoya City University
Curated by ChEMBL
Nagoya City University
Curated by ChEMBL
Affinity DataEC50: 940nMAssay Description:Agonist activity at human PPARdelta receptor expressed in HEK293 cells by GAL4 transactivation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+4nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at human GPR120-Galpha16 fusion protein expressed in Flp-in HEK293 cells assessed as effect on intracellular calcium concentration b...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Agonist activity at human GPR40 expressed in T-REx HEK293 cells assessed as effect on intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 86nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 159nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 2.61E+3nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 145nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 736nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 254nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 511nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 268nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 770nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 88nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 272nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 734nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 117nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 115nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 149nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 73nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 161nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 704nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 121nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 58nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 224nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 266nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Sanwa Kagaku Kenkyusho
Curated by ChEMBL
Affinity DataEC50: 331nMAssay Description:Agonist activity at mouse GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair