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Found 22 with Last Name = 'knapp' and Initial = 'ff'
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.0300nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.120nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.150nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKi:  0.160nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.260nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  0.270nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.760nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  0.780nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50456344(CHEMBL2112942)
Affinity DataKi:  1.10nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  5.20nMAssay Description:Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  28nMAssay Description:Ability to displace [3H]N-methylscopolamine (NMS) from M3 receptor in rat submaxillary gland homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  267nMAssay Description:Ability to displace [3H](-)-quinuclidinyl bezilate(QNB) from M2 receptor in rat heart homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  2.40nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  30nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKd:  0.200nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50450592(CHEMBL558910)
Affinity DataKd:  0.320nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50453895(CHEMBL2111842)
Affinity DataKd:  0.430nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Oak Ridge National Laboratory (Ornl)

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  0.356nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M4 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50453895(CHEMBL2111842)
Affinity DataKd:  0.230nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  6.80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  0.383nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M1 using [3H]QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Oak Ridge National Laboratory

Curated by ChEMBL
LigandPNGBDBM50031098((E)-(R)-2-Hydroxy-5-iodo-2-phenyl-pent-4-enoic aci...)
Affinity DataKd:  41nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M2 using [3H]-QNB as radioligand from rat heart tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed