Compile Data Set for Download or QSAR
maximum 50k data
Found 94 with Last Name = 'leroux' and Initial = 'v'
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206554(CHEMBL219777 | N-(4-fluoro-benzyl)-N'-hydroxy-2-[1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206558(CHEMBL375521 | N-hydroxy-N'-(4-phenyl-butyl)-2-[1-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206550(2-benzyl-N-hydroxy-N'-(2-methyl-benzyl)-malonamide...)
Affinity DataIC50:  41nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197503(CHEMBL425291 | N-hydroxy-2-isobutyl-N'-(3-phenoxy-...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197497(2-benzyl-N-hydroxy-N'-(4-phenyl-butyl)-malonamide ...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206556(2-Benzyl-N-(4-fluoro-benzyl)-N'-hydroxy-malonamide...)
Affinity DataIC50:  57nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197498(CHEMBL220311 | N-hydroxy-2-isobutyl-N'-(4-phenyl-b...)
Affinity DataIC50:  82nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206547(CHEMBL374479 | N-hydroxy-2-isobutyl-N'-naphthalen-...)
Affinity DataIC50:  91nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206543(2-benzyl-N-hydroxy-N'-naphthalen-1-ylmethyl-malona...)
Affinity DataIC50:  107nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206551(CHEMBL376198 | N-hydroxy-2-isobutyl-N'-(1,2,3,4-te...)
Affinity DataIC50:  109nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50062474(2,N-Dibenzyl-N'-hydroxy-malonamide | 2N-dibenzyl-N...)
Affinity DataIC50:  125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50062453(2-Benzyl-N-hydroxy-N'-(3-phenyl-propyl)-malonamide...)
Affinity DataIC50:  125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206552(2-(3-phenoxybenzyl)-N1-(4-chlorobenzyl)-N3-hydroxy...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)
Affinity DataIC50:  152nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197501(2-(3-phenoxybenzyl)-N1-benzyl-N3-hydroxymalonamide...)
Affinity DataIC50:  164nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206546(2-benzyl-N-(4-chloro-benzyl)-N'-hydroxy-malonamide...)
Affinity DataIC50:  170nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  171nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  206nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206557(2-benzyl-3-(4-benzyl-piperidin-1-yl)-N-hydroxy-3-o...)
Affinity DataIC50:  206nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197505(2-(3-phenoxybenzyl)-N1-hydroxy-N3-(4-phenylbutyl)m...)
Affinity DataIC50:  225nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50341636((3Z)-N-(3-CHLOROPHENYL)-3-({3,5-DIMETHYL-4-[(4-MET...)
Affinity DataIC50:  228nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206566(2-(3-phenoxybenzyl)-N1-(4-(trifluoromethyl)benzyl)...)
Affinity DataIC50:  231nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206564(2-(3-phenoxybenzyl)-3-(4-benzylpiperidin-1-yl)-N-h...)
Affinity DataIC50:  248nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206545(2-benzyl-3-(3,4-dihydro-1H-isoquinolin-2-yl)-N-hyd...)
Affinity DataIC50:  253nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  321nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206555(2-[1-Phenyl-meth-(Z)-ylidene]-malonic Acid Monoeth...)
Affinity DataIC50:  330nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197495(2-(4-benzyl-piperidine-1-carbonyl)-4-methyl-pentan...)
Affinity DataIC50:  406nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197503(CHEMBL425291 | N-hydroxy-2-isobutyl-N'-(3-phenoxy-...)
Affinity DataIC50:  443nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197503(CHEMBL425291 | N-hydroxy-2-isobutyl-N'-(3-phenoxy-...)
Affinity DataIC50:  443nMAssay Description:Inhibition of pig kidney microsomal APNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197495(2-(4-benzyl-piperidine-1-carbonyl)-4-methyl-pentan...)
Affinity DataIC50:  452nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197494(CHEMBL220253 | N-benzyl-N'-hydroxy-2-isobutyl-malo...)
Affinity DataIC50:  495nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206565(2-(3-phenoxybenzyl)-N1-hydroxy-N3-(3-phenylpropyl)...)
Affinity DataIC50:  527nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50062478(CHEMBL116641 | N-Hydroxy-2-isobutyl-N'-(3-phenyl-p...)
Affinity DataIC50:  528nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359983(CHEMBL1927769)
Affinity DataIC50:  559nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197494(CHEMBL220253 | N-benzyl-N'-hydroxy-2-isobutyl-malo...)
Affinity DataIC50:  590nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359984(CHEMBL1927768)
Affinity DataIC50:  607nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  620nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human HepG2 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197504(CHEMBL223711 | N1-benzyl-N3-hydroxy-2-((1-methyl-1...)
Affinity DataIC50:  718nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359985(CHEMBL1927772)
Affinity DataIC50:  760nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50062478(CHEMBL116641 | N-Hydroxy-2-isobutyl-N'-(3-phenyl-p...)
Affinity DataIC50:  790nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359986(CHEMBL1927625)
Affinity DataIC50:  793nMAssay Description:Inhibition of Met-mediated scattering in HGF-stimulated human MDCK cells pre-incubated overnight prior to HGF stimulation for 24 hrs measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359981(CHEMBL1927770)
Affinity DataIC50:  811nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197502(CHEMBL220010 | N-hydroxy-2-isobutyl-N'-phenethyl-m...)
Affinity DataIC50:  885nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197496(CHEMBL220176 | N-(4-chloro-benzyl)-N'-hydroxy-2-is...)
Affinity DataIC50:  904nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206553(2-(3-phenoxybenzyl)-3-(3,4-dihydroisoquinolin-2(1H...)
Affinity DataIC50:  966nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
University Of Lille 2

Curated by ChEMBL
LigandPNGBDBM50197502(CHEMBL220010 | N-hydroxy-2-isobutyl-N'-phenethyl-m...)
Affinity DataIC50:  984nMAssay Description:Inhibition of microsomal neural aminopeptidase in pig kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206544(2-benzyl-N-hydroxy-N'-phenethyl-malonamide | 2-ben...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50197498(CHEMBL220311 | N-hydroxy-2-isobutyl-N'-(4-phenyl-b...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50206548(2-benzyl-N-biphenyl-3-ylmethyl-N'-hydroxy-malonami...)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50359982(CHEMBL1927771)
Affinity DataIC50:  1.19E+3nMAssay Description:Inhibition of Met-mediated tumorigenesis in HGF-stimulated human GTL16 cells assessed as impairment in anchorage-independent growth by soft agar grow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 94 total ) | Next | Last >>
Jump to: