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Found 81 with Last Name = 'maschauer' and Initial = 's'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331552(CHEMBL1288585 | [11C]-(+)-(4aR,10bR)-4-propyl-3,4,...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50240845((S)-2-{(2S,3R)-2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Amin...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132057(CHEMBL1180430 | CHEMBL126128 | N-{4-[4-(2-Methoxy-...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132047(3-(4-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50443382(CHEMBL3086356)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM85050(CAS_184162-64-9 | SR 142948A | SR142948 | SR142948...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]neurotensin from human NTS1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331552(CHEMBL1288585 | [11C]-(+)-(4aR,10bR)-4-propyl-3,4,...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity to human dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132057(CHEMBL1180430 | CHEMBL126128 | N-{4-[4-(2-Methoxy-...)
Affinity DataKi:  13.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132047(3-(4-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  22.6nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]spiperone from human dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50184805(1-(2-methoxyphenyl)-4-((1-phenyl-1H-1,2,3-triazol-...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442747(CHEMBL2443009)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442750(CHEMBL2443006)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442752(CHEMBL2443004)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50184805(1-(2-methoxyphenyl)-4-((1-phenyl-1H-1,2,3-triazol-...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442751(CHEMBL2443005)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442750(CHEMBL2443006)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442746(CHEMBL2443010)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442748(CHEMBL2443008)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442749(CHEMBL2443007)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]SCH 23990 from dopamine D1 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(PIG)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50184805(1-(2-methoxyphenyl)-4-((1-phenyl-1H-1,2,3-triazol-...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442751(CHEMBL2443005)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442749(CHEMBL2443007)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442754(CHEMBL2443002)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442756(CHEMBL2443000)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442751(CHEMBL2443005)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442747(CHEMBL2443009)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442747(CHEMBL2443009)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442746(CHEMBL2443010)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442746(CHEMBL2443010)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442749(CHEMBL2443007)
Affinity DataKi:  770nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442747(CHEMBL2443009)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Sus scrofa)
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]SCH 23990 from dopamine D1 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442755(CHEMBL2443001)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442748(CHEMBL2443008)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442748(CHEMBL2443008)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442752(CHEMBL2443004)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442746(CHEMBL2443010)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Sus scrofa)
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50442753(CHEMBL2443003)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [3H]-prazosin from alpha1-adrenergic receptor in pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442750(CHEMBL2443006)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]spiperone from human D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442751(CHEMBL2443005)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-UniversitäT Erlangen-NüRnberg

Curated by ChEMBL
LigandPNGBDBM50442750(CHEMBL2443006)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]spiperone from human D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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