Affinity DataKi: 0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of [3H]PDBu binding to PKC alpha C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibition of [3H]PDBu binding to PKC delta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKC beta C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Inhibition of human GST-tagged 17betaHSD5 expressed in Escherichia coli by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]PDBu binding to PKC delta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of human AKR1C3 using S-(+)-1,2,3,4-tetrahydro-1-naphthol as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Inhibition of [3H]PDBu binding to PKC delta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]PDBu binding to PKC delta C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B peptideMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B peptideMore data for this Ligand-Target Pair